| Cell Based Assays for Drug Discovery ( )The | | | | 4. Strategic Analysis of the High-Content Tools |
| term drug discovery tools usually refers to | | | | Space 60 |
| high-content screening (HCS) and analysis and is | | | | 4.1 Analysis of the High-Content Market Structure |
| composed of those applications that require | | | | 60 |
| sufficient levels of sample throughput, whereby | | | | 4.2 Description of the Drug Discovery Marketplace |
| complex cellular events and phenotypes can be | | | | and Definition of the Field 60 |
| studied. | | | | 4.3 Key Market Drivers and Challenges in the |
| Elements of drug performance like toxicity and | | | | High-Content Analysis Space 61 |
| specificity can be established simultaneously using | | | | 4.4 Consolidated Picture of the High-Content |
| mixed cell types—primary cells, cell lines, cell | | | | Analysis Marketplace 65 |
| subpopulations. HCS seeks to assess the impact | | | | 4.5 High-Content Analysis Market Sectors and |
| of phenotypic and cellular changes that are | | | | Growth Rate 66 |
| brought about by gene modification (such as with | | | | 4.6 Vendors of High-Content Analysis Technology |
| RNA interference (RNAi) approaches) and/or drug | | | | 66 |
| (or compound) treatment. The purpose of this | | | | 5. High-Content Analysis Technology Platforms 67 |
| examination is to describe the specific segments | | | | 5.1 Methods of Digital Imaging 67 |
| of the global drug discovery tools market. Within | | | | 5.2 Fluorescence Microscopy 67 |
| this area, the report covers those segments that | | | | 5.3 Major High-Content Analysis Instrumentation |
| are highly active in terms of innovation and | | | | 68 |
| growth. Specifically, this study examines the | | | | 5.3.1 High-Content Analysis Platforms to Support |
| markets for small lab equipment all the way up to | | | | GPCR Screening 69 |
| highly automated, large automated platforms, as | | | | 5.4 High-Content Analysis Reagents 69 |
| well as accessory equipment such as reagents, | | | | 5.5 Imaging Software 70 |
| supplies and manufacturers’ original equipment | | | | 5.6 Enterprise-Level IT Solutions to Support |
| manufacturer (OEM) additional equipment. | | | | High-Content Screening Experiments 70 |
| Table of Contents: | | | | 5.6.1 Image Analysis Algorithms 71 |
| 1. Overview 5 | | | | 5.7 Use of RNAi in High-Content Analysis 73 |
| 1.1 Objectives of the Report 5 | | | | 5.8 Industry Alliances to Leverage RNAi and |
| 1.2 Methodology 6 | | | | High-Content Analysis 73 |
| 1.3 Scope of the Report 7 | | | | 5.9 Emerging Trends in High-Content Analysis |
| 1.4 Executive Summary 8 | | | | Technology Platforms 74 |
| 2. Technologies and Product Offering for | | | | 6. High-Content Analysis in Drug Selection, |
| High-Content Analysis 11 | | | | Screening and Biomarker Discovery 75 |
| 2.1 Definition of High-Content Analysis and Why it | | | | 6.1 Stem Cells as Tools for Drug Discovery 76 |
| is so Attractive a Discipline 12 | | | | 6.2 Cellular Systems Biology for Development of |
| 2.2 Classes of Measurements Possible with | | | | Toxicity Panels in Drug Safety Testing 76 |
| High-Content Analysis Approaches and Biological | | | | 6.3 Drug Discovery Companies Marketing |
| Functions Investigated 15 | | | | Cell-based Assays 77 |
| 2.3 Instrumentation Platforms for High-Content | | | | 6.4 Companies Using Cell-based Assays in Drug |
| Analysis 19 | | | | Discovery Programs 80 |
| 2.3.1 High-Content Screening Technology 19 | | | | 6.4.1 Phenotypic Drug Discovery (PDD) 80 |
| 2.4 Reagent and Assay Platforms for | | | | 6.4.2 Application of Quantitative High-Throughput |
| High-Content Analysis 26 | | | | Screening to HCA Cell-based Assays 80 |
| 2.5 Cell-based Screening Technologies in Drug | | | | 6.4.3 Application of High-Content Fingerprinting to |
| Development 29 | | | | Oncology Drug Discovery: Focus on in vitro and in |
| 2.5.1 Applications of Cell-based Assays 30 | | | | vivo Phenocopying and Cancer Stem Cell Analysis |
| 2.5.2 Pharma Drug Discovery Paradigm and | | | | 81 |
| Compound Screening 30 | | | | 6.5 Target Discovery and Validation by RNAi |
| 2.5.3 High-Content Analysis in the | | | | Screening 81 |
| Biopharmaceutical Industry 31 | | | | 6.6 FLIM-FRET Methodology 81 |
| 3. Market Analysis of the High-Content Tools | | | | 6.7 Multidimensional Fluorescence Imaging (MDFI) |
| Space 33 | | | | Technology 81 |
| 3.1 High-Content Analysis Market Size and Growth | | | | 7. Company Profiles 82 |
| 33 | | | | 7.1 Acumen Pharmaceuticals, Inc. 82 |
| 3.2 Market Survey to Assess Qualitative and | | | | 7.2 Acumen Bioscience (division of TTP Group) 82 |
| Quantitative Parameters of the High-Content | | | | 7.3 Applied Biosystems 82 |
| Analysis Space 33 | | | | 7.4 BD Biosciences 84 |
| 3.3 Experimental and Research Trends in | | | | 7.5 DiscoveRX 84 |
| High-Content Analysis 35 | | | | 7.6 Evotec Technologies (acquired by PerkinElmer) |
| 3.4 Challenges and Market Drivers in High-Content | | | | 84 |
| Analysis 40 | | | | 7.7 Fisher BioImage 84 |
| 3.4.1 Barriers to High-Content Analysis 42 | | | | 7.8 General Electric, GE Healthcare 85 |
| 3.4.2 Drivers of High-Content Analysis 43 | | | | 7.9 Guava Technologies (now a division of Millipore) |
| 3.5 High-Content Analysis in Combination with RNAi | | | | 85 |
| 43 | | | | 7.10 Integral Molecular (Akceli Inc.) 86 |
| 3.6 Market Landscape of Instrumentation for | | | | 7.11 LemnaTech GmbH 86 |
| High-Content Analysis 45 | | | | 7.12 Millipore 86 |
| 3.7 Reagent and Assay Usage in High-Content | | | | 7.13 Molecular Devices Corporation, now a division |
| Analysis 49 | | | | of MDS Analytical Techniques 88 |
| 3.8 Trends in the High-Content Analysis Assays | | | | 7.14 NIH Chemical Genomics Center 90 |
| Reagents Space—Major Product Vendors 52 | | | | 7.15 PerkinElmer 91 |
| 3.9 Emerging Market Trends in High-Content | | | | 7.16 Sangamo Biosciences, Inc. 93 |
| Analysis 54 | | | | 7.17 Spotfire (acquired by TIBCO) 93 |
| 3.10 Market Forecasts for the High-Content | | | | 7.18 Thermo Scientific Cellomics 94 |
| Analysis Space 57 | | | | 7.19 Translational Genomics Research Institute 94 |
| 3.11 Use of HCS in Pharmaceutical Companies 58 | | | | 7.20 Vala Sciences, Inc. 94 |
| 3.12 Qualitative Opportunities and Challenges for | | | | 8. |
| Market Adoption 59 | | | | |